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Last Update 11/25/2010
2010
Original Papers

Convergent assembly of the spiroacetal subunit of didemnaketal B.
H. Fuwa, S. Noji, and M. Sasaki
Org. Lett., 12, 5354-5357 (2010).

An enantioselective total synthesis of aspergillides A and B.
H. Fuwa, H. Yamaguchi, and M. Sasaki
Tetrahedron, 66, 7492-7503 (2010).

Studies toward the total synthesis of gambieric acids: Stereocontrolled synthesis of a DEFG-ring model compound.
H. Fuwa, S. Noji, and M. Sasaki
J. Org. Chem., 75, 5072-5082 (2010).
Most Read Articles ranked #17 (July 2010)

A concise total synthesis of (+/-)-centrolobine.
H. Fuwa, K. Noto, and M. Sasaki
Heterocycles, 82 (Dr. Albert Eschenmoser special issue) , in press (2010).

The marine polyether gambierol enhances muscle contraction and blocks a transient K+ current in skeletal muscle cells.
S. Schulmberger, G. Ouanounou, E. Girard, M. Sasaki, H. Fuwa, M. C. Louzao, L. M. Botana, E. Benoit, and J. Molgo
Toxicon, 56, 785-791 (2010).

Improved synthesis and in vitro/in vivo activities of natural product-inspired, artificial glutamate analogs.
M. Oikawa, M. Ikoma, M. Sasaki, M. B. Gill, G. T. Swanson, K. Shimamoto, and R. Sakai
Bioorg. Med. Chem., 18, 3795-3804 (2010).

A unified total synthesis of aspergillides A and B.
H. Fuwa, H. Yamaguchi, and M. Sasaki.
Org. Lett., 12, 1848-1851 (2010).

Most Read Articles ranked #10 (March 2010)

Stereoselective synthesis of substituted tetrahydropyrans via domino olefin cross-metathesis/intramolecular oxa-conjugate cyclization.
H. Fuwa, K. Noto, and M. Sasaki.
Org. Lett., 12, 1636-1639 (2010).

An efficient synthesis of 2,6-disubstituted 2,3-dihydro-4H-pyran-4-ones via Sonogashira coupling of p-toluenethiol esters
H. Fuwa, S. Matsukida, and M. Sasaki
Synlett, 1239-1242 (2010).

Highlighted in SYNFACTS, 1239 (2010).

A series of structurally novel heterotricyclic a-amino-3-hydroxyl-5-methyl-4-isooxazole-propionate receptor-selective antagonists
M. B. Gill, S. Frausto, M. Ikoma, M. Sasaki, M. Oikawa, R. Sakai, and G. T. Swanson.
Br. J. Pharmacol., 159, 1417-1429 (2010).

A concise total synthesis of (+)-neopeltolide.
H. Fuwa, A. Saito, and M. Sasaki.
Angew. Chem., Int. Ed., 49, 3041-3044 (2010).

Most Accessed Articles ranked #10 (March 2010)

Calcium oscillations induced by gambierol in cerebellar granule cells
E. Alonso, C. Vale, M. Sasaki, H. Fuwa, Y. Konno, S. Perez, M. R. Vieytes, L. M. Botana.
J. Cell. Biochem., 110, 497-508 (2010).

Total synthesis of (-)-exiguolide
H. Fuwa and M. Sasaki.
Org. Lett., 12, 584-587 (2010).

Most Read Articles ranked #2 (January 2010)
Most Accessed Articles 2010 ranked #3 (throughout 2010)

Pharmacological activity of C10-substituted analogs of the high-affinity kainate receptor agonist dysiherbaine
L. L. Lash-Van Wyhe, P. A. Postila, K. Tsubone, M. Sasaki, O. T. Pentikainen, R. Sakai, and G. T. Swanson
Neuropharmacol., 58, 640-649 (2010).

Highly efficient synthesis of medium-sized lactones via oxidative lactonization: Concise total synthesis of isolaurepan
M. Ebine, Y. Suga, H. Fuwa, and M. Sasaki.
Org. Biomol. Chem., 8, 39-42 (2010).

Top 10 Most Accessed Articles ranked #2 (December 2009)

Reviews and Accounts

Total synthesis of structurally complex marine oxacyclic natural products.
H. Fuwa
Bull. Chem. Soc. Jpn. (Award Account), 83, 1401-1420 (2010).

著書
理科年表(国立天文台編、丸善)
佐々木 誠 編集
平成22年度 生体物質 物182−物193、生理活性物質195−199.

Copyright(C) Sasaki Group 2009