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Last Update 11/12/2014
Original Papers

Effect of gambierol and its heptacyclic and tetracyclic analogues in cultured cerebellar neurons. A structure-activity relationships study.
S. Perez, C. Vale, E. Alonso, H. Fuwa, M. Sasaki, Y. Konno, T. Goto, Y. Suga, M. R. Vieytes, L. M. Botana
Chem. Res. Toxicol., 25, 1929-1937 (2012).

Tandem catalysis in domino olefin cross-metathesis/intramolecular oxa-conjugate cyclization: Concise synthesis of 2,6-cis-substituted tetrahydropyran derivatives
H. Fuwa, T. Noguchi, K. Noto, M. Sasaki
Org. Biomol. Chem., 10, 8108-8112 (2012).

Total synthesis and complete stereostructure of gambieric acid A
H. Fuwa, K. Ishigai, K. Hashizume, M. Sasaki
J. Am. Chem. Soc., 134, 11984-11987 (2012).
Most Read Articles in July 2012
Highlighted in SYNFACTS, 8, 1053 (2012)

A concise synthesis of the AB-ring fragment of (-)-gambierol
H. Fuwa, K. Hirota, M. Sasaki
Heterocycles, 86 (Professor Ei-ichi Negishi special issue), 127-132 (2012).
This paper was written on invitation.

Stereoselective synthesis of the C1-C16 fragment of goniodomin A
M. Nakajima, H. Fuwa, M. Sasaki
Bull. Chem. Soc. Jpn., 85, 948-956 (2012).
Selected Papers of the September 2012 issue of BCSJ

Total synthesis of (-)-polycavernoside A: Suzuki-Miyaura coupling approach
Y. Kasai, T. Ito, M. Sasaki
Org. Lett., 14, 3186-3189 (2012).
Most Read Articles in June 2012

Design and synthesis of skeletal analogues of gambierol: Attenuation of amyloid-b and tau pathology with voltage-gated potassium channel and N-methyl-D-aspartate receptor implications
E. Alonso, H. Fuwa, C. Vale, Y. Suga, T. Goto, Y. Konno, M. Sasaki, F. M. LaFerla, M. R. Vieytes, L. Gimenez-Llort, L. M. Botana
J. Am. Chem. Soc., 134, 7467-7479 (2012).

Stereoselective synthesis of 2,6-cis-substituted tetrahydropyrans: Bronsted acid-catalyzed intramolecular oxa-conjugate cyclization of a,b-unsaturated ester surrogates
H. Fuwa, N. Ichinokawa, K. Noto, and M. Sasaki
J. Org. Chem., 77, 2588-2607 (2012).

This paper was selected as a Featured Article of The Journal of Organic Chemistry.
This paper was featured in the Front Cover of The Journal of Organic Chemistry.

Reviews and Accounts

Total synthesis of tetrahydropyran-containing natural products exploiting intramolecular oxa-conjugate cyclization
H. Fuwa
Heterocycles, 85, 1255-1298 (2012).
This review was written on invitation.


トップドラッグから学ぶ創薬化学 有機合成化学協会編(東京化学同人)、p. 140, 158, 159 (2012)

理科年表 平成25年(国立天文台編、丸善)
佐々木 誠 編集
生体物質 物182−物193、生理活性物質195−199.

Copyright(C) Sasaki Group 2012